Enantioselective synthesis of aspergillide B.
نویسندگان
چکیده
The enantioselective synthesis of aspergillide B, a 14-membered macrocyclic cytotoxin, was achieved in a 49% yield via 7 steps from a synthetic intermediate of aspergillide C. The spectroscopic data and specific rotation value for the synthetic material matched those of natural aspergillide B.
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ورودعنوان ژورنال:
- Bioscience, biotechnology, and biochemistry
دوره 73 8 شماره
صفحات -
تاریخ انتشار 2009